PF 03716556 ( —— )

产品货号. M16652 CAS No. 928774-43-0

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

PF 03716556
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

PF 3716556 is a potent and selective P-CAB (potassium-competitive acid blocker), with pIC50 of 6.026 and 7.095 for the inhibition of porcine H+,K+-ATPase activity in ion-leaky and ion-tight assay, respectively.
产品描述

PF 3716556 is a potent and selective P-CAB (potassium-competitive acid blocker), with pIC50 of 6.026 and 7.095 for the inhibition of porcine H+,K+-ATPase activity in ion-leaky and ion-tight assay, respectively, inhibits gastric acid secretion, displays no activity at Na+,K+-ATPase, used for the treatment of gastroesophageal reflux disease.
同义词

——
通路

Endocrinology/Hormones
靶点

ATPase
受体

H+/K+-ATPase
研究领域

Metabolic Disease
适应症

——

1.Mori, et al. J Pharmacol Exp Ther. 2009 Feb;328(2):671-9.

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